Publicaciones en las que colabora con Antonio Ferrer Montiel (12)

2023

  1. β-Lactam TRPM8 Antagonists Derived from Phe-Phenylalaninol Conjugates: Structure–Activity Relationships and Antiallodynic Activity

    International Journal of Molecular Sciences, Vol. 24, Núm. 19

2022

  1. β-Lactam TRPM8 Antagonist RGM8-51 Displays Antinociceptive Activity in Different Animal Models

    International Journal of Molecular Sciences, Vol. 23, Núm. 5

2021

  1. A capsaicinoid-based soft drug, AG1529, for attenuating TRPV1-mediated histaminergic and inflammatory sensory neuron excitability

    Scientific Reports, Vol. 11, Núm. 1

  2. DD04107-Derived neuronal exocytosis inhibitor peptides: Evidences for synaptotagmin-1 as a putative target

    Bioorganic Chemistry, Vol. 115

2020

  1. Highly functionalized β-lactams and 2-ketopiperazines as TRPM8 antagonists with antiallodynic activity

    Scientific Reports, Vol. 10, Núm. 1

  2. Structure-Based Design of Novel Biphenyl Amide Antagonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 8 Channels with Potential Implications in the Treatment of Sensory Neuropathies

    ACS Chemical Neuroscience, Vol. 11, Núm. 3, pp. 268-290

2019

  1. 1-(2′,5′-Dihydroxyphenyl)-3-(2-fluoro-4-hydroxyphenyl)-1-propanone (RGM079): A Positive Allosteric Modulator of α7 Nicotinic Receptors with Analgesic and Neuroprotective Activity

    ACS Chemical Neuroscience, Vol. 10, Núm. 8, pp. 3900-3909

2018

  1. Amino acid and peptide prodrugs of diphenylpropanones positive allosteric modulators of α7 nicotinic receptors with analgesic activity

    European Journal of Medicinal Chemistry, Vol. 143, pp. 157-165

  2. Identification of a Potent Tryptophan-Based TRPM8 Antagonist with in Vivo Analgesic Activity

    Journal of Medicinal Chemistry, Vol. 61, Núm. 14, pp. 6140-6152

  3. TRP channels as potential targets for sex-related differences in migraine pain

    Frontiers in Molecular Biosciences, Vol. 5, Núm. AUG

  4. Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders

    Journal of Medicinal Chemistry, Vol. 61, Núm. 10, pp. 4436-4455

2012

  1. An inhibitor of neuronal exocytosis (DD04107) displays long-lasting in vivo activity against chronic inflammatory and neuropathic pain

    Journal of Pharmacology and Experimental Therapeutics, Vol. 341, Núm. 3, pp. 634-645