FARMACOLOGÍA DEL DOLOR EXPERIMENTAL
FARMADEX
Antonio
Ferrer Montiel
Publications by the researcher in collaboration with Antonio Ferrer Montiel (12)
2023
-
β-Lactam TRPM8 Antagonists Derived from Phe-Phenylalaninol Conjugates: Structure–Activity Relationships and Antiallodynic Activity
International Journal of Molecular Sciences, Vol. 24, Núm. 19
2022
-
β-Lactam TRPM8 Antagonist RGM8-51 Displays Antinociceptive Activity in Different Animal Models
International Journal of Molecular Sciences, Vol. 23, Núm. 5
2021
-
A capsaicinoid-based soft drug, AG1529, for attenuating TRPV1-mediated histaminergic and inflammatory sensory neuron excitability
Scientific Reports, Vol. 11, Núm. 1
-
DD04107-Derived neuronal exocytosis inhibitor peptides: Evidences for synaptotagmin-1 as a putative target
Bioorganic Chemistry, Vol. 115
2020
-
Highly functionalized β-lactams and 2-ketopiperazines as TRPM8 antagonists with antiallodynic activity
Scientific Reports, Vol. 10, Núm. 1
-
Structure-Based Design of Novel Biphenyl Amide Antagonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 8 Channels with Potential Implications in the Treatment of Sensory Neuropathies
ACS Chemical Neuroscience, Vol. 11, Núm. 3, pp. 268-290
2019
-
1-(2′,5′-Dihydroxyphenyl)-3-(2-fluoro-4-hydroxyphenyl)-1-propanone (RGM079): A Positive Allosteric Modulator of α7 Nicotinic Receptors with Analgesic and Neuroprotective Activity
ACS Chemical Neuroscience, Vol. 10, Núm. 8, pp. 3900-3909
2018
-
Amino acid and peptide prodrugs of diphenylpropanones positive allosteric modulators of α7 nicotinic receptors with analgesic activity
European Journal of Medicinal Chemistry, Vol. 143, pp. 157-165
-
Identification of a Potent Tryptophan-Based TRPM8 Antagonist with in Vivo Analgesic Activity
Journal of Medicinal Chemistry, Vol. 61, Núm. 14, pp. 6140-6152
-
TRP channels as potential targets for sex-related differences in migraine pain
Frontiers in Molecular Biosciences, Vol. 5, Núm. AUG
-
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders
Journal of Medicinal Chemistry, Vol. 61, Núm. 10, pp. 4436-4455
2012
-
An inhibitor of neuronal exocytosis (DD04107) displays long-lasting in vivo activity against chronic inflammatory and neuropathic pain
Journal of Pharmacology and Experimental Therapeutics, Vol. 341, Núm. 3, pp. 634-645