Medicina
Departament
Instituto de Química Médica
Madrid, EspañaPublicacions en col·laboració amb investigadors/es de Instituto de Química Médica (7)
2023
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β-Lactam TRPM8 Antagonists Derived from Phe-Phenylalaninol Conjugates: Structure–Activity Relationships and Antiallodynic Activity
International Journal of Molecular Sciences, Vol. 24, Núm. 19
2022
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β-Lactam TRPM8 Antagonist RGM8-51 Displays Antinociceptive Activity in Different Animal Models
International Journal of Molecular Sciences, Vol. 23, Núm. 5
2021
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DD04107-Derived neuronal exocytosis inhibitor peptides: Evidences for synaptotagmin-1 as a putative target
Bioorganic Chemistry, Vol. 115
2020
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Highly functionalized β-lactams and 2-ketopiperazines as TRPM8 antagonists with antiallodynic activity
Scientific Reports, Vol. 10, Núm. 1
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New cannabinoid receptor antagonists as pharmacological tool
Bioorganic and Medicinal Chemistry, Vol. 28, Núm. 19
2019
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1-(2′,5′-Dihydroxyphenyl)-3-(2-fluoro-4-hydroxyphenyl)-1-propanone (RGM079): A Positive Allosteric Modulator of α7 Nicotinic Receptors with Analgesic and Neuroprotective Activity
ACS Chemical Neuroscience, Vol. 10, Núm. 8, pp. 3900-3909
2018
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Amino acid and peptide prodrugs of diphenylpropanones positive allosteric modulators of α7 nicotinic receptors with analgesic activity
European Journal of Medicinal Chemistry, Vol. 143, pp. 157-165