Publications in collaboration with researchers from KU Leuven (12)

2023

  1. Convergent Approaches and Biological Activity of C1 and/or C3 Mono or Diamino Derivatives of 1α,25-Dihydroxy-19-nor-vitamin D3. Key Enzymatic Desymmetrization of A-Ring Synthon Precursor

    Advanced Synthesis and Catalysis, Vol. 365, Núm. 2, pp. 201-210

2018

  1. Enzymatic Desymmetrization of 19-nor-Vitamin D3 A-Ring Synthon Precursor: Synthesis, Structure Elucidation, and Biological Activity of 1α,25-Dihydroxy-3-epi-19-nor-vitamin D3 and 1β,25-Dihydroxy-19-nor-vitamin D3

    Advanced Synthesis and Catalysis, Vol. 360, Núm. 14, pp. 2762-2772

2017

  1. A-Ring-Modified 2-Hydroxyethylidene Previtamin D3Analogues: Synthesis and Biological Evaluation

    European Journal of Organic Chemistry, Vol. 2017, Núm. 3, pp. 504-513

2009

  1. Synthesis, conformational analysis, and biological evaluation of 19-nor-vitamin D3 analogues with A-ring modifications

    Journal of Medicinal Chemistry, Vol. 52, Núm. 19, pp. 6158-6162

2008

  1. Synthesis and biological activity of previtamin D3 analogues with A-ring modifications

    Bioorganic and Medicinal Chemistry, Vol. 16, Núm. 24, pp. 10244-10250

2007

  1. Synthesis and biological evaluation of new 6-s-cis locked 1,2,25-trihydroxyprevitamin D3 analogues

    Bioorganic and Medicinal Chemistry, Vol. 15, Núm. 12, pp. 4193-4202

2006

  1. Novel A-ring homodimeric C-3-carbamate analogues of 1α,25-dihydroxyvitamin D3: Synthesis and preliminary biological evaluation

    Bioorganic and Medicinal Chemistry, Vol. 14, Núm. 22, pp. 7512-7519

  2. Versatile synthesis and biological evaluation of 1,3-diamino-substituted 1α,25-dihydroxyvitamin D3 analogues

    Bioorganic and Medicinal Chemistry, Vol. 14, Núm. 4, pp. 928-937

2004

  1. Chemoenzymatic syntheses of homo- and heterodimers of AZT and d4T, and evaluation of their anti-HIV Activity

    Nucleosides, Nucleotides and Nucleic Acids, Vol. 23, Núm. 4, pp. 701-714

  2. Chemoenzymatic synthesis and biological evaluation of C-3 carbamate analogues of 1α,25-dihydroxyvitamin D 3

    Bioorganic and Medicinal Chemistry, Vol. 12, Núm. 20, pp. 5443-5451

2003

  1. Synthesis and antiviral activity assay of novel (E)-3′,5′ -diamino-5-(2-bromovinyl)-2′,3′,5′-trideoxyuridine

    Nucleosides, Nucleotides and Nucleic Acids

  2. Synthesis, protonation behavior, conformational analysis, and regioselective enzymatic acylation of the novel diamino analogue of (E)-5-(2-bromovinyl)-2′-deoxyuridine (BVDU)

    Nucleosides, Nucleotides and Nucleic Acids, Vol. 22, Núm. 10, pp. 1939-1952