FARMADEX
Farmacología del Dolor Experimental
Publications (3) Publications in which a researcher has participated
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Drug Discovery
2023
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β-Lactam TRPM8 Antagonists Derived from Phe-Phenylalaninol Conjugates: Structure–Activity Relationships and Antiallodynic Activity
International Journal of Molecular Sciences, Vol. 24, Núm. 19
2020
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Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities
Journal of Medicinal Chemistry, Vol. 63, Núm. 17, pp. 9672-9694
2019
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1-(2′,5′-Dihydroxyphenyl)-3-(2-fluoro-4-hydroxyphenyl)-1-propanone (RGM079): A Positive Allosteric Modulator of α7 Nicotinic Receptors with Analgesic and Neuroprotective Activity
ACS Chemical Neuroscience, Vol. 10, Núm. 8, pp. 3900-3909